Macitentan, ≥99%

Catalog No. 040588

General Information

Synonyms	ACT-064992
CAS No.	441798-33-0
M.F.	C₁₉H₂₀Br₂N₆O₄S
M.W.	588.27
MDL No.	MFCD17167076

Technical Data

Appearance	White to off-white crystalline powder
Assay	≥99% HPLC
Solubility	DMSO
Storage	-20℃
Description	Macitentana is an orally active, non-peptide, dual ETA/ETB (endothelin) receptor antagonist with IC50 of 0.5 nM/391 nM.

Reference

Corallo C, et al. J Biol Regul Homeost Agents. 2013 Apr-Jun;27(2):455-62
Bruderer S, et al. Pharmacology. 2013;91(5-6):331-8
Atsmon J, et al. Clin Pharmacokinet. 2013 Aug;52(8):685-92
Weiss J, et al. Eur J Pharmacol. 2013 Feb 15;701(1-3):168-75
Kim SJ, et al. Transl Oncol. 2012 Feb;5(1):39-47

Size	Price	Quantity	Favorites
10 mg	USD290
50 mg	USD725

Please inquire for non-standard packs and bulk quantities.

Availability: Ships in 4 days

For research use only. Not for human use.

> Certificate of Analysis

> MSDS

	(*Required Field)
*Name
*Organization Name
*Country
*Email Address
Phone
Subject	040588, Macitentan, ≥99%, 441798-33-0
*Message
*Code

Macitentan, ≥99%

Inquire