Giacomini, K.M., et al. Nat. Rev. Drug Discov. 9, 215-236, (2010)
Knütter, I., et al. J. Pharmacol. Exp. Ther. 327, 432-441, (2008)
Maurin, C., et al. J. Med. Chem., 47, 5583 (2004)
Marchand, C., et al. Mol. Pharmacol., 64, 600 (2003)
Subissi, A., et al. Cardivascular Drug Reviews, 17, 2 (1999)
Gorren, A., et al. Biochem. J., 331, 801 (1998)
DeForrest, J.M., et al. J. Cardiovasc. Pharmacol. 13, 887-894, (1989)